the correlations between chemical structure properties and antiviral activities of hiv-1 inhibitors: the study of anti-aids

Authors

majid monajjemi

anita abedib

abstract

in this work, we calculated the several physico chemical properties containing of solubility (byvcl), lipophilicity (by milinspiration), dipole and quadrupole moments (by density functionaltheory) for 7 azt analogs, and compared these parameters with inhibition assays of them. it isresulted; cytotoxicity of these drugs is related with their lipophilicity inversely. with using of thisresult, for 7 nucleoside analoges we predict, cytotoxicity addition arrangement are as following:cbv> d4t> ddi> azt> ddc> abc> 3tc

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Journal title:
journal of physical & theoretical chemistry

ISSN

volume 1

issue 4 2005

Keywords
[ ' h i v ' , 1 , ' c y t o t o x i c i t y ' , ' l i p o p h i l i c i t y ' , ' s o l u b i l i t y ' , ' m o m e n t s ' ]

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